SCHEMBL18322969

SCHEMBL18322969

O=CN1CCC(Oc2ccc(-c3ccc4ccccc4n3)cc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.50
RAB9A P51151 6/20 0.50
KDM4E B2RXH2 4/20 0.50
SMN1; SMN2 Q16637 4/20 0.50
ALDH1A1 P00352 2/20 0.50
NFKB1 P19838 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPT P10636 3/20 0.46
CYP3A4 P08684 3/20 0.46
GMNN O75496 1/20 0.46
TP53 P04637 1/20 0.46
PKM P14618 1/20 0.46
HPGD P15428 1/20 0.46
THPO P40225 1/20 0.46
BLM P54132 1/20 0.46
PMP22 Q01453 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18322889 0.84 NPC1 (0.44) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL18319055 0.81 MAPT (0.48) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL18322884 0.81 NPC1 (0.50) NPC1RAB9ASMN1; SMN2CYP3A4HRH3
SCHEMBL18318517 0.80 NAMPT (0.49) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL18318563 0.80 NPC1 (0.47) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL30497909 0.79 CA12 (0.44) CYP3A4HRH3KCNH2ADRA1AFASN
SCHEMBL18318859 0.79 CA12 (0.44) CYP3A4HRH3KCNH2ADRA1AFASN
Hydrochloric Acid SCHEMBL28550768 0.78 CA12 (0.43) CYP3A4HRH3KCNH2ADRA1AFASN
SCHEMBL18318037 0.76 NAMPT (0.56) KDM4EALDH1A1KMT2AMAPTGAA
SCHEMBL18318038 0.76 NAMPT (0.56) KDM4EALDH1A1KMT2AMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3310441-A1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES Cephalon, Inc. (US) 2018-04-25 EP disclosed
WO-2016205633-A1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON, INC. (US) 2016-12-22 WO disclosed