Diphosphomelavonate

Diphosphomelavonate

SCHEMBL183248

CC(O)(CCOP(=O)(O)OP(=O)(O)O)CC(=O)O

nearest known ligand 0.64

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MVD P53602 4/20 0.64
HMGCR P04035 1/20 0.44
CHRM1 P11229 1/20 0.44
TBXA2R P21731 1/20 0.44
ADRA1A P35348 1/20 0.44
BTN3A1 O00481 3/20 0.44
FFAR1 O14842 1/20 0.35
CPT2 P23786 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
FNTA P49354 2/20 0.33
FNTB P49356 2/20 0.33
GGPS1 O95749 2/20 0.32
PGGT1B P53609 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diphosphomelavonate SCHEMBL3272270 1.00 MVD (0.64) MVDHMGCRCHRM1TBXA2RADRA1A
Diphosphomelavonate SCHEMBL29398109 1.00 MVD (0.64) MVDHMGCRCHRM1TBXA2RADRA1A
SCHEMBL599363 0.86 HMGCR (0.50) MVDHMGCRCHRM1TBXA2RADRA1A
SCHEMBL1286788 0.86 HMGCR (0.50) MVDHMGCRCHRM1TBXA2RADRA1A
SCHEMBL18376075 0.86 HMGCR (0.50) MVDHMGCRCHRM1TBXA2RADRA1A
SCHEMBL15258419 0.85 MVD (0.47) MVDHMGCRCHRM1TBXA2RADRA1A
SCHEMBL14864445 0.84 MVD (0.47) MVDHMGCRCHRM1TBXA2RADRA1A
SCHEMBL18281294 0.84 MVD (0.51) MVDHMGCRCHRM1TBXA2RADRA1A
SCHEMBL1995374 0.83 BTN3A1 (0.55) MVDHMGCRCHRM1TBXA2RADRA1A
Isopentenylpyrophosphate SCHEMBL10944407 0.81 BTN3A1 (0.61) MVDHMGCRCHRM1TBXA2RADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 514 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114480242-B Escherichia coli engineering bacteria for MK-n production and construction method thereof 中国科学院合肥物质科学研究院 2023-04-25 CN claimed
CN-112391327-B Engineering bacterium for co-production of geraniol and nerol and construction method and application thereof 中国农业科学院烟草研究所 2022-08-05 CN claimed
CN-114480242-A Escherichia coli engineering bacterium for MK-n production and construction method thereof 中国科学院合肥物质科学研究院 2022-05-13 CN claimed
EP-2764084-B2 UTILIZATION OF PHOSPHOKETOLASE IN THE PRODUCTION OF MEVALONATE, ISOPRENOID PRECURSORS, AND ISOPRENE DANISCO US INC (US) 2021-11-03 EP claimed
CN-113151340-A Genetic engineering bacterium for increasing yield of beta-carotene and application thereof 广州智特奇生物科技股份有限公司 2021-07-23 CN claimed
US-20210071150-A1 METHOD FOR INCREASING THE YIELD OF OXIDOSQUALENE, TRITERPENES AND/OR TRITERPENOIDS AND HOST CELL THEREFORE WESTFAELISCHE WILHELMS-UNIVERSITAET MUENSTER (DE) 2021-03-11 US claimed
EP-3775181-A1 METHOD FOR INCREASING THE YIELD OF OXIDOSQUALENE, TRITERPENES AND/OR TRITERPENOIDS AND HOST CELL THEREFORE Fraunhofer Gesellschaft zur Förderung der Angewand (DE) 2021-02-17 EP claimed
EP-3107993-B1 RECOMBINANT MICROORGANISMS FOR THE ENHANCED PRODUCTION OF MEVALONATE, ISOPRENE, ISOPRENOID PRECURSORS, ISOPRENOIDS, AND ACETYL-COA-DERIVED PRODUCTS DANISCO US INC (US) 2020-08-26 EP claimed
EP-3368673-B1 COMPOSITIONS AND METHODS FOR PRODUCTION OF MYRCENE AMYRIS INC (US) 2020-07-29 EP claimed
US-20200129579-A1 METHOD FOR REPAIRING SKIN DAMAGE CAUSED BY PARTICULATE MATTERS (PMs) SHANGHAI ZHONGYI DAILY CHEMICAL CO., LTD. (CN) 2020-04-30 US claimed
WO-2019197327-A1 METHOD FOR INCREASING THE YIELD OF OXIDOSQUALENE, TRITERPENES AND/OR TRITERPENOIDS AND HOST CELL THEREFORE FRAUNHOFER-GESELLSCHAFT ZUR FOERDERUNG DER ANGEWANDTEN FORSCHUNG E.V. (DE) 2019-10-17 WO claimed
EP-2971027-B1 USE OF PHOSPHOKETOLASE AND PHOSPHOTRANSACETYLASE FOR PRODUCTION OF ACETYL-COENZYME A DERIVED COMPOUNDS AMYRIS INC (US) 2019-01-30 EP claimed
EP-2764084-B1 UTILIZATION OF PHOSPHOKETOLASE IN THE PRODUCTION OF MEVALONATE, ISOPRENOID PRECURSORS, AND ISOPRENE DANISCO US INC (US) 2018-02-28 EP claimed
EP-2776571-B1 PRODUCTION OF ACETYL-COENZYME A DERIVED ISOPRENOIDS AMYRIS INC (US) 2017-04-12 EP claimed
EP-2875136-B1 RHODOBACTER FOR PREPARING TERPENOIDS ISOBIONICS B V (NL) 2017-04-12 EP claimed
EP-2707475-B1 PRODUCTION OF ACETYL-COENZYME A DERIVED COMPOUNDS AMYRIS INC (US) 2015-09-30 EP claimed
EP-1947189-A2 Method of vitamin production DCV Inc. doing business as Bio-Technical Resourses (US) 2008-07-23 EP claimed
US-20070254354-A1 Production of Isoprenoids Amyris, Inc. 2007-11-01 US claimed
WO-2001077366-A1 POSITIVE SELECTION METHOD, COMPOUNDS, HOST CELLS AND USES THEREOF CUBIST PHARMACEUTICALS, INC. (US) 2001-10-18 WO claimed
WO-1995013058-A1 HALOGENATED MEVALONATE COMPOSITIONS AND USES THEREOF IN RAS-DEPENDENT CELL GROWTH BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1995-05-18 WO claimed