SCHEMBL18340752

SCHEMBL18340752

CN(C)C/C=C/CNc1ccc(C(=O)Nc2ccc(Nc3cc(-c4cnc5c(ccn5S(=O)(=O)c5ccccc5)c4)ncn3)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIP4K2A P48426 14/20 0.54
PIP4K2B P78356 14/20 0.54
PIP4K2C Q8TBX8 1/20 0.42
PIKFYVE Q9Y2I7 1/20 0.42
EGFR P00533 1/20 0.39
ERBB2 P04626 1/20 0.39
ERBB4 Q15303 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
MAPK8 P45983 2/20 0.37
MAPK9 P45984 2/20 0.37
CDK7 P50613 2/20 0.36
CCNH P51946 2/20 0.36
MAPK10 P53779 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18340698 0.96 PIP4K2A (0.57) PIP4K2APIP4K2BPIP4K2CPIKFYVEMAPK8
SCHEMBL18340763 0.94 PIP4K2A (0.57) PIP4K2APIP4K2BPIP4K2CPIKFYVEEGFR
SCHEMBL29888558 0.92 PIP4K2A (0.65) PIP4K2APIP4K2BPIP4K2CPIKFYVEEGFR
SCHEMBL20093356 0.92 PIP4K2A (0.65) PIP4K2APIP4K2BPIP4K2CPIKFYVEEGFR
SCHEMBL18340738 0.91 PIP4K2A (0.56) PIP4K2APIP4K2BPIP4K2CPIKFYVEEGFR
SCHEMBL20093361 0.88 PIP4K2A (0.68) PIP4K2APIP4K2BPIP4K2CPIKFYVEMAPK8
SCHEMBL18340701 0.87 PIP4K2A (0.47) PIP4K2APIP4K2BPIP4K2CPIKFYVEMAPK8
SCHEMBL20093369 0.86 PIP4K2A (0.67) PIP4K2APIP4K2BPIP4K2CPIKFYVEEGFR
SCHEMBL18340771 0.85 MAPK8 (0.44) PIP4K2APIP4K2BEGFRERBB2ERBB4
SCHEMBL18340750 0.85 PIP4K2A (0.43) PIP4K2APIP4K2BPIP4K2CEGFRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3313530-A1 4,6-PYRIMIDINYLENE DERIVATIVES AND USES THEREOF Dana Farber Cancer Institute, Inc. (US) 2018-05-02 EP disclosed
WO-2016210296-A1 4,6-PYRIMIDINYLENE DERIVATIVES AND USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2016-12-29 WO disclosed