SCHEMBL1835672

SCHEMBL1835672

Cc1ccccc1-c1cccc(C)c1C(=O)N1CCCC(Nc2ccc(C(F)(F)F)cn2)C1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 1/20 0.50
HCRTR1 O43613 15/20 0.47
HCRTR2 O43614 8/20 0.47
CCR5 P51681 1/20 0.45
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1835677 0.87 KDM4E (0.52) MAP3K12HCRTR1HCRTR2
SCHEMBL1835674 0.84 MAP3K12 (0.49) MAP3K12HCRTR1HCRTR2KMT2A
SCHEMBL20144969 0.82 HCRTR1 (0.64) HCRTR1HCRTR2
SCHEMBL20145041 0.82 HCRTR1 (0.64) HCRTR1HCRTR2
SCHEMBL1141302 0.82 MAP3K12 (0.51) MAP3K12HCRTR1HCRTR2
SCHEMBL1141304 0.82 MAP3K12 (0.51) MAP3K12HCRTR1HCRTR2
SCHEMBL18697648 0.81 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL20144838 0.81 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL20144954 0.79 HCRTR1 (0.67) HCRTR1HCRTR2
SCHEMBL20144938 0.79 HCRTR1 (0.66) MAP3K12HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318367-A1 PIPERIDINE AND PYRROLIDINE COMPOUNDS Actelion Pharmaceuticals Ltd. (CH) 2011-05-11 EP disclosed