SCHEMBL18376752

SCHEMBL18376752

COc1ccc(-c2cccc3cnc(Nc4ccc(N5CCOCC5)nc4)nc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTK P33981 1/20 0.56
MAPK10 P53779 7/20 0.54
JUN P05412 5/20 0.54
MAPK8 P45983 5/20 0.54
KDM4E B2RXH2 1/20 0.53
GAA P10253 1/20 0.53
CSF1R P07333 1/20 0.53
DAPK1 P53355 1/20 0.53
KCNH2 Q12809 1/20 0.53
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MTOR P42345 1/20 0.48
SMG1 Q96Q15 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
FGFR2 P21802 1/20 0.47
FGFR3 P22607 1/20 0.47
ZAP70 P43403 1/20 0.47
CDK1 P06493 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29205095 0.95 MAPK10 (0.55) TTKMAPK10JUNMAPK8KDM4E
SCHEMBL30859690 0.95 MAPK10 (0.55) TTKMAPK10JUNMAPK8KDM4E
SCHEMBL18376760 0.90 TTK (0.66) TTKMAPK10JUNMAPK8CSF1R
SCHEMBL29848408 0.88 MAPK10 (0.66) TTKMAPK10JUNMAPK8DGAT1
SCHEMBL16514447 0.88 MAPK10 (0.66) TTKMAPK10JUNMAPK8DGAT1
SCHEMBL16514209 0.87 MAPK10 (0.49) TTKMAPK10JUNMAPK8CSF1R
SCHEMBL16514195 0.87 MAPK10 (0.50) TTKMAPK10JUNMAPK8NPC1
SCHEMBL1632167 0.86 MAPK10 (0.57) TTKMAPK10JUNMAPK8MTOR
SCHEMBL18376252 0.85 TTK (0.65) TTKMAPK10JUNMAPK8NPC1
SCHEMBL30859695 0.85 TTK (0.65) TTKMAPK10JUNMAPK8NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017005137-A1 QUINAZOLINE COMPOUND, INTERMEDIATE, PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USES THEREOF 吉林大学 2017-01-12 WO disclosed