SCHEMBL18436105

SCHEMBL18436105

CCC(=O)N1C(C)CN(c2ccc(-c3cnc4c(-c5ccc(C#N)cc5)cccc4c3O)cn2)CC1C

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.43
CHRM2 P08172 1/20 0.39
PARP1 P09874 5/20 0.38
PARP2 Q9UGN5 4/20 0.38
KDM4A O75164 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
SMO Q99835 3/20 0.37
HRH4 Q9H3N8 1/20 0.36
EGLN1 Q9GZT9 3/20 0.36
CNR2 P34972 1/20 0.36
KRAS P01116 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
RET P07949 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17128172 1.00 CHRM1 (0.43) CHRM1CHRM2PARP1PARP2KDM4A
SCHEMBL17128173 0.90 CHRM1 (0.42) CHRM1CHRM2PARP1PARP2HRH4
SCHEMBL18436684 0.90 CHRM1 (0.42) CHRM1CHRM2PARP1PARP2HRH4
SCHEMBL21336707 0.89 CNR2 (0.37) CHRM1SMOCNR2
SCHEMBL17128122 0.84 CHRM1 (0.42) CHRM1CHRM2PARP1PARP2HRH4
SCHEMBL18420369 0.84 CHRM1 (0.42) CHRM1CHRM2PARP1PARP2HRH4
SCHEMBL21336763 0.84 CHRM1 (0.42) CHRM1CHRM2PARP1PARP2HRH4
SCHEMBL18420409 0.83 CHRM1 (0.43) CHRM1CHRM2PARP1PARP2SMO
SCHEMBL17127936 0.83 CHRM1 (0.43) CHRM1CHRM2PARP1PARP2SMO
SCHEMBL18436392 0.82 CHRM1 (0.42) CHRM1CHRM2PARP1PARP2HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed