SCHEMBL18436110

SCHEMBL18436110

CC(C)(O)c1ccc(N2CCNCC2=O)nc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.39
HRH3 Q9Y5N1 1/20 0.38
OGA O60502 1/20 0.38
SMO Q99835 1/20 0.37
TNKS O95271 1/20 0.37
PARP1 P09874 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
OPRD1 P41143 1/20 0.36
EED O75530 1/20 0.35
SUZ12 Q15022 1/20 0.35
EZH2 Q15910 1/20 0.35
PRMT5 O14744 1/20 0.35
MAPT P10636 4/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
APAF1 O14727 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TLR8 Q9NR97 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29977962 1.00 PIM1 (0.39) PIM1HRH3OGASMOTNKS
Hydrochloric Acid SCHEMBL29978429 0.99 PIM1 (0.39) PIM1HRH3OGASMOTNKS
Hydrochloric Acid SCHEMBL28343839 0.99 PIM1 (0.39) PIM1HRH3OGASMOTNKS
SCHEMBL1578382 0.84 MAPT (0.48) PIM1MAPTALDH1A1KDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL1962520 0.83 MAPT (0.47) PIM1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL1578400 0.79 BPTF (0.43) PIM1EEDSUZ12EZH2PRMT5
SCHEMBL18740364 0.79 PIM1 (0.42) PIM1PARP1EEDSUZ12EZH2
Hydrochloric Acid SCHEMBL1964613 0.78 BPTF (0.42) PIM1EEDSUZ12EZH2PRMT5
Hydrochloric Acid SCHEMBL28662945 0.78 PIM1 (0.42) PIM1PARP1EEDSUZ12EZH2
SCHEMBL17128345 0.77 OGA (0.50) HRH3OGASMOOPRD1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110494431-B Azacyclo derivative, preparation method and medical application thereof 苏州浦合医药科技有限公司 2022-11-04 CN disclosed
CN-110494431-A Nitrogen heterocycles derivative, preparation method and its medical usage BEIJING YUEZHIKANGTAI BIOMEDICINES CO LTD 2019-11-22 CN disclosed
EP-3124482-B1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO LTD (CN) 2019-09-11 EP disclosed
WO-2019062657-A1 NITROGEN HETEROCYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 北京越之康泰生物医药科技有限公司 2019-04-04 WO disclosed
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed