SCHEMBL18436126

SCHEMBL18436126

COC(=O)N1C(C)CN(c2ccc(-c3cnc4c(-c5ccc(C#N)cc5)cccc4c3OC)cc2)CC1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
KIT P10721 2/20 0.36
JAK1 P23458 1/20 0.36
SLC22A12 Q96S37 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
NR3C2 P08235 1/20 0.34
PTPN11 Q06124 1/20 0.34
MAPKAPK2 P49137 2/20 0.34
TGFBR1 P36897 1/20 0.34
ACVR1 Q04771 1/20 0.34
JAK2 O60674 1/20 0.34
CHRM4 P08173 2/20 0.34
GRIA2 P42262 1/20 0.34
KCNH2 Q12809 1/20 0.34
EGLN1 Q9GZT9 2/20 0.33
PRKDC P78527 1/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
HTR7 P34969 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21336923 1.00 CHRM2 (0.37) CHRM2HRH4KITJAK1SLC22A12
SCHEMBL17127783 1.00 CHRM2 (0.37) CHRM2HRH4KITJAK1SLC22A12
SCHEMBL18436341 1.00 CHRM2 (0.37) CHRM2HRH4KITJAK1SLC22A12
SCHEMBL17128117 0.93 MEN1 (0.38) CHRM2HRH4JAK1MAPKAPK2TGFBR1
SCHEMBL18436078 0.92 CHRM2 (0.39) CHRM2HRH4KITEGLN1
SCHEMBL17128175 0.92 CHRM2 (0.39) CHRM2HRH4KITEGLN1
SCHEMBL17128386 0.92 CHRM2 (0.39) CHRM2HRH4KITEGLN1
SCHEMBL18436834 0.92 CHRM2 (0.39) CHRM2HRH4KITEGLN1
SCHEMBL17128119 0.90 CHRM2 (0.34) CHRM2HRH4KITJAK1SLC22A12
SCHEMBL17128014 0.90 CHRM2 (0.36) CHRM2HRH4KITJAK1SLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed