SCHEMBL18436556

SCHEMBL18436556

c1ccc(N2CC3CC2CO3)cc1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 1/20 0.45
SYK P43405 1/20 0.43
PDE10A Q9Y233 1/20 0.41
MAP3K12 Q12852 8/20 0.40
MTOR P42345 2/20 0.40
PIK3CA P42336 1/20 0.40
SOS1 Q07889 1/20 0.36
MAP3K13 O43283 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21256819 0.82 SOS1 (0.39) PRKDCMAP3K12MTORPIK3CASOS1
SCHEMBL12082429 0.82 SOS1 (0.39) PRKDCMAP3K12MTORPIK3CASOS1
SCHEMBL21256815 0.82 SOS1 (0.39) PRKDCMAP3K12MTORPIK3CASOS1
SCHEMBL15399039 0.82 MAP3K12 (0.44) PRKDCMAP3K12MTORPIK3CASOS1
SCHEMBL25889732 0.82 MAP3K12 (0.39) PRKDCSYKPDE10AMAP3K12MTOR
SCHEMBL20448663 0.82 MAP3K12 (0.39) PRKDCSYKPDE10AMAP3K12MTOR
SCHEMBL25889731 0.82 MAP3K12 (0.39) PRKDCSYKPDE10AMAP3K12MTOR
SCHEMBL23387212 0.77 NSD2 (0.42) PRKDC
SCHEMBL19221692 0.76 MAPT (0.41) PRKDC
SCHEMBL23707037 0.73 MAP3K12 (0.43) MAP3K12MTORPIK3CAMAP3K13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-B1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO LTD (CN) 2019-09-11 EP disclosed
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed