SCHEMBL18436662

SCHEMBL18436662

O=[N+]([O-])Sc1cccc(OCc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 6/20 0.56
MAOA P21397 2/20 0.56
TLR4 O00206 1/20 0.56
TLR2 O60603 1/20 0.56
NR4A2 P43354 1/20 0.50
CYP4F2 P78329 1/20 0.48
CYP4A11 Q02928 1/20 0.48
BCHE P06276 1/20 0.48
PTPN1 P18031 1/20 0.47
GRM5 P41594 1/20 0.46
CCNB2 O95067 1/20 0.46
CDK1 P06493 1/20 0.46
CDK4 P11802 1/20 0.46
CCNB1 P14635 1/20 0.46
CCND1 P24385 1/20 0.46
CCNB3 Q8WWL7 1/20 0.46
SMPD1 P17405 1/20 0.46
ALOX5 P09917 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13596117 0.80 MAOB (0.54) MAOBMAOATLR4TLR2ALDH1A1
SCHEMBL3175420 0.79 MAOB (0.61) MAOBMAOANR4A2CYP4F2CYP4A11
SCHEMBL2965418 0.77 MAOB (0.63) MAOBMAOATLR4TLR2ALDH1A1
SCHEMBL11742933 0.77 MAOB (0.59) MAOBMAOATLR4TLR2NR4A2
SCHEMBL30443578 0.77 MAOB (0.63) MAOBMAOATLR4TLR2ALDH1A1
SCHEMBL11566779 0.76 MAOB (0.62) MAOBMAOANR4A2CYP4F2CYP4A11
SCHEMBL11566776 0.76 MAOB (0.57) MAOBMAOANR4A2CYP4F2CYP4A11
SCHEMBL4411578 0.76 PDE7A (0.51) MAOBMAOATLR4TLR2NR4A2
SCHEMBL31187444 0.75 SPHK2 (0.59) MAOBMAOANR4A2CYP4F2CYP4A11
SCHEMBL1268719 0.75 MAOB (0.81) MAOBMAOANR4A2CYP4F2CYP4A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2511262-B1 PROCESS FOR PRODUCING 2-AMINO-2-[2-[4-(3-BENZYLOXY-PHENYLTHIO)-2-CHLOROPHENYL[ETHYL]-1,3-PROPANEDIOL HYDROCHLORIDE KYORIN SEIYAKU KK (JP) 2017-02-01 EP disclosed