SCHEMBL18436982

SCHEMBL18436982

CCC(=O)N1[C@@H]2CC[C@H]1CN(c1ccc(SC)cn1)C2

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.42
HDAC1 Q13547 2/20 0.38
JAK2 O60674 11/20 0.38
JAK1 P23458 11/20 0.38
TYK2 P29597 11/20 0.38
CHRM1 P11229 1/20 0.37
RET P07949 1/20 0.37
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
SLC6A4 P31645 1/20 0.36
HTR7 P34969 1/20 0.36
DRD3 P35462 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18436009 0.84 PDE10A (0.43) HDAC1JAK2JAK1TYK2CHRM1
SCHEMBL18435972 0.84 PDE10A (0.43) HDAC1JAK2JAK1TYK2CHRM1
SCHEMBL17128204 0.82 JAK2 (0.41) ACACBHDAC1JAK2JAK1TYK2
SCHEMBL17128199 0.82 ACACB (0.43) ACACBHDAC1JAK2JAK1TYK2
SCHEMBL19012542 0.82 HDAC1 (0.41) HDAC1JAK2JAK1TYK2CHRM1
SCHEMBL19012547 0.81 ACACB (0.47) ACACBHDAC1JAK2JAK1TYK2
SCHEMBL19001048 0.81 HPGD (0.42) HDAC1JAK2JAK1TYK2CHRM1
SCHEMBL20034304 0.81 ACACB (0.47) ACACBHDAC1JAK2JAK1TYK2
SCHEMBL19001060 0.81 HPGD (0.42) HDAC1JAK2JAK1TYK2CHRM1
SCHEMBL19001192 0.78 ACACB (0.40) ACACBHDAC1JAK2JAK1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed