SCHEMBL1844827

SCHEMBL1844827

O=C(COCc1ccccc1)NC1CC(n2cnc3c(NCC(c4ccccc4)c4ccccc4)nc(Cl)nc32)C(O)C1O

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 13/20 0.57
ADORA3 P0DMS8 10/20 0.56
ADORA1 P30542 2/20 0.52
NT5E P21589 4/20 0.48
TMIGD3 P0DMS9 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
HTR3A P46098 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL242820 1.00 ADORA2A (0.57) ADORA2AADORA3ADORA1NT5ETMIGD3
SCHEMBL1401984 0.91 ADORA2A (0.67) ADORA2AADORA3ADORA1NT5E
SCHEMBL1412472 0.89 ADORA2A (0.55) ADORA2AADORA3ADORA1NT5E
SCHEMBL3118651 0.89 ADORA2A (0.55) ADORA2AADORA3ADORA1NT5E
SCHEMBL1412375 0.89 ADORA2A (0.55) ADORA2AADORA3ADORA1NT5E
SCHEMBL241285 0.89 ADORA2A (0.58) ADORA2AADORA3ADORA1NT5E
SCHEMBL1401973 0.89 ADORA2A (0.69) ADORA2AADORA3ADORA1NT5E
SCHEMBL241132 0.88 ADORA2A (0.60) ADORA2AADORA3ADORA1
SCHEMBL1412152 0.88 ADORA2A (0.70) ADORA2AADORA3ADORA1
SCHEMBL1412300 0.88 ADORA2A (0.70) ADORA2AADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2322525-A1 Purine derivatives for use as adenosin A2A receptor agonists Novartis AG (CH) 2011-05-18 EP disclosed