SCHEMBL18480656

SCHEMBL18480656

COc1cc(OC)c(/C=C/S(=O)(=O)Cc2ccc(OC)c(NS(C)(=O)=O)c2)c(OC)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 4/20 0.70
MET P08581 1/20 0.70
NQO2 P16083 1/20 0.70
FECH P22830 1/20 0.70
CLK3 P49761 1/20 0.70
HDAC3 O15379 2/20 0.67
HDAC4 P56524 2/20 0.67
HDAC1 Q13547 2/20 0.67
HDAC7 Q8WUI4 2/20 0.67
HDAC2 Q92769 2/20 0.67
HDAC10 Q969S8 2/20 0.67
HDAC11 Q96DB2 2/20 0.67
HDAC8 Q9BY41 2/20 0.67
HDAC6 Q9UBN7 2/20 0.67
HDAC9 Q9UKV0 2/20 0.67
HDAC5 Q9UQL6 2/20 0.67
MAPK1 P28482 2/20 0.44
ALDH1A1 P00352 1/20 0.44
PTK2B Q14289 1/20 0.44
PTK2 Q05397 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1122953 0.88 PLK1 (0.72) PLK1METNQO2FECHCLK3
SCHEMBL1122955 0.88 PLK1 (0.72) PLK1METNQO2FECHCLK3
SCHEMBL18437835 0.88 PLK1 (0.66) PLK1METNQO2FECHCLK3
SCHEMBL1123384 0.88 PLK1 (0.66) PLK1METNQO2FECHCLK3
SCHEMBL1123194 0.88 PLK1 (0.66) PLK1METNQO2FECHCLK3
SCHEMBL18437833 0.88 PLK1 (0.66) PLK1METNQO2FECHCLK3
SCHEMBL18481195 0.87 PLK1 (0.69) PLK1METNQO2FECHCLK3
SCHEMBL12132322 0.87 PLK1 (0.66) PLK1METNQO2FECHCLK3
SCHEMBL16366467 0.86 PLK1 (0.74) PLK1METNQO2FECHCLK3
SCHEMBL15835693 0.86 PLK1 (0.77) PLK1METNQO2FECHCLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017023912-A1 2,4,6-TRIALKOXYSTRYL ARYL SULFONES, SULFONAMIDES AND CARBOXAMIDES, AND METHODS OF PREPARATION AND USE TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2017-02-09 WO disclosed