SCHEMBL18509710

SCHEMBL18509710

Cc1c(CCC(=O)O)c2cccc(N)c2n1C

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
PARP1 P09874 1/20 0.43
HDAC6 Q9UBN7 1/20 0.40
CMA1 P23946 1/20 0.40
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.39
FABP4 P15090 3/20 0.39
FABP5 Q01469 3/20 0.39
FABP3 P05413 1/20 0.39
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
CYSLTR2 Q9NS75 3/20 0.38
CYSLTR1 Q9Y271 3/20 0.38
PLA2G4A P47712 1/20 0.37
KDM4E B2RXH2 1/20 0.37
TBXAS1 P24557 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19872770 0.86 EGFR (0.48) EGFRNPC1RAB9AHDAC6CMA1
SCHEMBL21392209 0.86 EGFR (0.49) EGFRNPC1RAB9APARP1HDAC6
SCHEMBL20120013 0.83 EGFR (0.46) EGFRNPC1RAB9AGAACYSLTR2
SCHEMBL21392207 0.83 EGFR (0.46) EGFRNPC1RAB9AHDAC6CMA1
SCHEMBL18509698 0.83 EGFR (0.46) EGFRNPC1RAB9AHDAC6CMA1
SCHEMBL18509922 0.81 EGFR (0.47) EGFRNPC1RAB9AHDAC6CMA1
SCHEMBL18509747 0.81 EGFR (0.47) EGFRNPC1RAB9AHDAC6CMA1
SCHEMBL18509551 0.81 ABCB1 (0.48) EGFRNPC1RAB9AALDH1A1GAA
SCHEMBL18509744 0.80 EGFR (0.43) EGFRNPC1RAB9AHDAC6CMA1
SCHEMBL18509286 0.79 SLC22A12 (0.42) EGFRNPC1RAB9AHDAC6CMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081456-A1 HIGHLY ACTIVE SELF-SUFFICIENT NITRATION BIOCATALYSTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2018-05-03 WO disclosed
WO-2016134145-A9 ARTIFICIAL SELF-SUFFICIENT CYTOCHROME P450S UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2017-02-16 WO disclosed