SCHEMBL18524809

SCHEMBL18524809

CC(C)(C)NC(=O)Oc1c[nH]c2ncc(-c3nn(CC4CCNC4)c4ccc(OC(F)F)cc34)nc12

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SYK P43405 20/20 0.66
KCNH2 Q12809 6/20 0.66
CYP2D6 P10635 3/20 0.66
CYP2C9 P11712 3/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18524691 0.95 SYK (0.68) SYKKCNH2CYP2D6CYP2C9
SCHEMBL18524684 0.94 SYK (0.70) SYKKCNH2CYP2D6CYP2C9
SCHEMBL18524747 0.91 SYK (0.80) SYKKCNH2CYP2D6CYP2C9
SCHEMBL14737741 0.89 SYK (0.82) SYKKCNH2CYP2D6CYP2C9
SCHEMBL18524518 0.88 SYK (0.59) SYKKCNH2CYP2D6CYP2C9
SCHEMBL18524623 0.85 SYK (0.66) SYKKCNH2CYP2D6CYP2C9
SCHEMBL18524542 0.85 SYK (0.69) SYKKCNH2CYP2D6CYP2C9
SCHEMBL18524637 0.85 SYK (0.68) SYKKCNH2CYP2D6CYP2C9
SCHEMBL18524607 0.85 SYK (0.60) SYKKCNH2CYP2D6CYP2C9
SCHEMBL18524833 0.84 SYK (0.65) SYKKCNH2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2763990-B1 PYRROLOPYRAZINE KINASE INHIBITORS HOFFMANN LA ROCHE (CH) 2017-02-22 EP claimed