SCHEMBL18534372

SCHEMBL18534372

C=Cc1cc2c(cc1Sc1nc3c(N)ncnc3n1CCNCC(C)(C)C)OCC2

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 19/20 0.61
HSP90AB1 P08238 10/20 0.56
ERBB2 P04626 1/20 0.54
CDC37 Q16543 1/20 0.48
TRAP1 Q12931 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18534329 0.92 HSP90AA1 (0.69) HSP90AA1HSP90AB1ERBB2CDC37TRAP1
SCHEMBL11985173 0.89 HSP90AA1 (0.59) HSP90AA1HSP90AB1ERBB2CDC37TRAP1
SCHEMBL21442809 0.89 HSP90AA1 (0.76) HSP90AA1HSP90AB1ERBB2CDC37TRAP1
SCHEMBL1669635 0.88 HSP90AB1 (0.64) HSP90AA1HSP90AB1ERBB2CDC37TRAP1
SCHEMBL15980491 0.88 HSP90AA1 (0.56) HSP90AA1HSP90AB1ERBB2CDC37TRAP1
SCHEMBL15980479 0.88 HSP90AA1 (0.56) HSP90AA1HSP90AB1ERBB2CDC37TRAP1
SCHEMBL19265055 0.88 HSP90AB1 (0.54) HSP90AA1HSP90AB1ERBB2TRAP1
SCHEMBL17715305 0.88 HSP90AA1 (0.60) HSP90AA1HSP90AB1ERBB2CDC37TRAP1
SCHEMBL21442789 0.87 HSP90AA1 (0.80) HSP90AA1HSP90AB1CDC37TRAP1
SCHEMBL1672118 0.86 HSP90AA1 (0.54) HSP90AA1HSP90AB1ERBB2CDC37TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3208615-B1 USES OF LABELED HSP90 INHIBITORS SLOAN KETTERING INST CANCER RES (US) 2019-10-09 EP disclosed
EP-2729806-B1 USES OF LABELED HSP90 INHIBITORS SLOAN-KETTERING INST FOR CANCER RES (US) 2017-02-22 EP disclosed