SCHEMBL18534997

SCHEMBL18534997

Cn1ccc2ccnc(Br)c21

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CB P42338 1/20 0.34
MAPT P10636 1/20 0.34
SCN9A Q15858 1/20 0.31
LPO P22079 1/20 0.30
CDK4 P11802 1/20 0.30
CCND1 P24385 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19117686 0.78 CYP2A6 (0.41) PIK3CBMAPTSCN9A
SCHEMBL29942174 0.76 RXFP1 (0.35) PIK3CBMAPTSCN9ALPO
SCHEMBL22863238 0.76 PIK3CB (0.34) PIK3CBMAPTSCN9ALPO
SCHEMBL20987529 0.76 PIK3CB (0.38) PIK3CBMAPTSCN9ALPO
SCHEMBL3570930 0.76 RXFP1 (0.35) PIK3CBMAPTSCN9ALPO
SCHEMBL23346951 0.76 PIK3CB (0.42) PIK3CBMAPT
SCHEMBL29777078 0.76 PIK3CB (0.34) PIK3CBMAPTSCN9ALPO
SCHEMBL22863378 0.73 MAPT (0.40) PIK3CBMAPTSCN9ACDK4CCND1
SCHEMBL30122603 0.73 RXFP1 (0.33) PIK3CBMAPTSCN9A
SCHEMBL19759422 0.73 HASPIN (0.33) PIK3CBMAPTSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2763990-B1 PYRROLOPYRAZINE KINASE INHIBITORS HOFFMANN LA ROCHE (CH) 2017-02-22 EP disclosed