SCHEMBL1854853

SCHEMBL1854853

CCCCc1oc2ccccc2c1CN

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 11/20 0.58
EYA3 Q99504 2/20 0.50
TTR P02766 1/20 0.46
KDM4A O75164 1/20 0.45
KDM5A P29375 1/20 0.45
ING2 Q9H160 1/20 0.45
THRA P10827 1/20 0.43
THRB P10828 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1853311 0.98 PTPN1 (0.56) PTPN1EYA3TTRKDM4AKDM5A
SCHEMBL2985777 0.95 PTPN1 (0.53) PTPN1EYA3TTRKDM4AKDM5A
SCHEMBL8810393 0.84 PTPN1 (0.61) PTPN1EYA3TTRTHRATHRB
SCHEMBL11218137 0.83 PTPN1 (0.57) PTPN1EYA3TTR
Hydrochloric Acid SCHEMBL8732680 0.83 PTPN1 (0.60) PTPN1EYA3TTRTHRATHRB
SCHEMBL13049676 0.78 PTPN1 (0.55) PTPN1EYA3TTRTHRATHRB
SCHEMBL21555485 0.78 PTPN1 (0.52) PTPN1EYA3TTR
SCHEMBL6718612 0.78 PTPN1 (0.56) PTPN1EYA3TTRTHRATHRB
SCHEMBL11402772 0.78 PTPN1 (0.50) PTPN1EYA3
SCHEMBL24026894 0.77 PTPN1 (0.51) PTPN1EYA3TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1470102-B1 SUBSTITUTED METHYLENE AMIDE DERIVATIVES AS MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPS) MERCK SERONO SA (CH) 2011-05-25 EP disclosed