SCHEMBL18567412

SCHEMBL18567412

CC1(C)SC[C@@](C)(c2sc(-c3nnc(-c4ccc(F)cc4)o3)cc2Cl)NC1=N

nearest known ligand 0.52

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.52
BACE2 Q9Y5Z0 14/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18567410 0.92 BACE1 (0.51) BACE1BACE2
SCHEMBL18567769 0.90 BACE1 (0.51) BACE1BACE2
SCHEMBL18567766 0.90 BACE1 (0.53) BACE1BACE2
SCHEMBL18567411 0.89 BACE1 (0.54) BACE1BACE2
SCHEMBL18567775 0.86 BACE1 (0.54) BACE1BACE2
SCHEMBL15693514 0.83 BACE1 (0.65) BACE1BACE2
SCHEMBL17127261 0.79 BACE1 (0.66) BACE1BACE2
SCHEMBL20056278 0.77 BACE1 (0.51) BACE1BACE2
SCHEMBL15693515 0.75 BACE1 (0.64) BACE1BACE2
SCHEMBL15693516 0.74 BACE1 (0.55) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697210-B1 5-SUBSTITUTED IMINOTHIAZINES AND THEIR MONO-AND DIOXIDES AS BACE INHIBITORS, COMPOSITIONS, AND THEIR USE MERCK SHARP & DOHME (US) 2017-03-01 EP disclosed