SCHEMBL18598010

SCHEMBL18598010

CC1OCC2(c3cc(N)ccc3F)N=C(N)SCC12

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.57
BACE2 Q9Y5Z0 7/20 0.49
CTSD P07339 2/20 0.49
KCNH2 Q12809 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11326483 1.00 BACE1 (0.57) BACE1BACE2CTSDKCNH2
SCHEMBL11886481 0.90 BACE1 (0.48) BACE1BACE2CTSDKCNH2
SCHEMBL15986167 0.89 BACE1 (0.59) BACE1BACE2CTSDKCNH2
SCHEMBL11888116 0.87 BACE1 (0.51) BACE1BACE2CTSDKCNH2
SCHEMBL20341373 0.87 BACE1 (0.62) BACE1BACE2CTSD
SCHEMBL18011791 0.87 BACE1 (0.62) BACE1BACE2CTSD
SCHEMBL11028559 0.86 BACE1 (0.62) BACE1BACE2CTSD
SCHEMBL15986391 0.86 BACE1 (0.53) BACE1BACE2CTSDKCNH2
SCHEMBL2622844 0.86 BACE1 (0.59) BACE1BACE2CTSDKCNH2
SCHEMBL11888095 0.86 BACE1 (0.59) BACE1BACE2CTSDKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2665716-B1 METHODS AND COMPOUNDS USEFUL IN THE SYNTHESIS OF FUSED AMINODIHYDROTHIAZINE DERIVATIVES EISAI R&D MAN CO LTD (JP) 2017-03-08 EP disclosed