SCHEMBL1859907

SCHEMBL1859907

CC(C)(C)OC(=O)N1C[C@H](O)C[C@H]1C(=O)Nc1c(C(N)=O)oc2ccc(Br)cc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.51
POLB P06746 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 4/20 0.43
MAPT P10636 2/20 0.43
MEN1 O00255 3/20 0.42
ABL1 P00519 2/20 0.39
BCR P11274 2/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
TSHR P16473 3/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
USP30 Q70CQ3 1/20 0.38
HTRA1 Q92743 1/20 0.38
BACE1 P56817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1852387 1.00 CYP1A2 (0.51) CYP1A2POLBCYP3A4CYP2C19KMT2A
SCHEMBL1852389 1.00 CYP1A2 (0.51) CYP1A2POLBCYP3A4CYP2C19KMT2A
SCHEMBL1855450 0.91 KMT2A (0.43) CYP1A2POLBCYP3A4CYP2C19KMT2A
SCHEMBL1855448 0.91 KMT2A (0.43) CYP1A2POLBCYP3A4CYP2C19KMT2A
SCHEMBL1856586 0.91 KMT2A (0.43) CYP1A2POLBCYP3A4CYP2C19KMT2A
SCHEMBL1856064 0.90 KDM4E (0.52) CYP1A2POLBCYP3A4CYP2C19KMT2A
SCHEMBL1856066 0.90 KDM4E (0.52) CYP1A2POLBCYP3A4CYP2C19KMT2A
SCHEMBL1854752 0.87 USP30 (0.47) KMT2AMAPTMEN1ALDH1A1KDM4E
SCHEMBL1851649 0.87 USP30 (0.47) KMT2AMAPTMEN1ALDH1A1KDM4E
SCHEMBL4273196 0.86 KMT2A (0.44) KMT2AMAPTMEN1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097419-B1 BENZOFUROPYRIMIDINONES AS PROTEIN KINASE INHIBITORS EXELIXIS INC (US) 2011-05-25 EP disclosed