SCHEMBL18600005

SCHEMBL18600005

Nc1ccc(-c2nc(C(=O)Nc3cnccc3N3CCNCC3)cs2)cc1

nearest known ligand 0.76

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 20/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14328604 0.93 CHEK1 (0.81) CHEK1
SCHEMBL14328599 0.91 CHEK1 (0.77) CHEK1
SCHEMBL13156153 0.90 CHEK1 (0.85) CHEK1
SCHEMBL14206552 0.89 CHEK1 (0.74) CHEK1
SCHEMBL18600041 0.88 CHEK1 (0.86) CHEK1
SCHEMBL14206544 0.88 CHEK1 (0.79) CHEK1
SCHEMBL14206447 0.88 CHEK1 (0.73) CHEK1
SCHEMBL14328791 0.88 CHEK1 (0.72) CHEK1
SCHEMBL14328465 0.87 CHEK1 (0.72) CHEK1
SCHEMBL14206566 0.87 CHEK1 (1.00) CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078003-B1 ANILINOPIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF MERCK SHARP & DOHME (US) 2017-03-08 EP disclosed