SCHEMBL18601786

SCHEMBL18601786

CCN(CC)C(=O)CCCC(=O)c1cccc(CN2CN(c3ccccc3)C3(CCN(C(=O)OC(C)(C)C)CC3)C2=O)c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.51
TP53 P04637 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
MAPT P10636 1/20 0.51
ALOX15 P16050 1/20 0.51
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
NPC1L1 Q9UHC9 5/20 0.50
DDR1 Q08345 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL319273 0.88 NPC1L1 (0.51) MEN1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL318225 0.85 NPC1L1 (0.59) MEN1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL10248363 0.84 NPC1L1 (0.58) MEN1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL320092 0.83 NPC1L1 (0.57) MEN1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL318110 0.82 NPC1L1 (0.55) MEN1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL5563023 0.82 NPC1L1 (0.64) NPC1L1DDR1
SCHEMBL9998932 0.81 NPC1L1 (0.52) MEN1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL318941 0.81 NPC1L1 (0.52) MEN1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL318940 0.81 NPC1L1 (0.52) MEN1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL9999126 0.80 NPC1L1 (0.52) MEN1TP53CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3138841-A1 D2 ANTAGONISTS, METHODS OF SYNTHESIS AND METHODS OF USE Altos Therapeutics, LLC (US) 2017-03-08 EP disclosed