SCHEMBL18607247

SCHEMBL18607247

CC(F)Oc1cc(N2CCC(N(C)C)CC2)c(N)cc1Nc1nccc(-c2noc3ccccc23)n1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LCK P06239 2/20 0.47
EGFR P00533 12/20 0.42
ALK Q9UM73 4/20 0.41
CDK4 P11802 2/20 0.34
CCNA2 P20248 2/20 0.34
CCND1 P24385 2/20 0.34
CDK2 P24941 2/20 0.34
CCNA1 P78396 2/20 0.34
GSK3B P49841 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18607248 0.95 LCK (0.48) LCKEGFRALK
SCHEMBL18607249 0.95 LCK (0.48) LCKEGFRALK
SCHEMBL18606892 0.91 LCK (0.51) LCKEGFR
SCHEMBL18607244 0.88 LCK (0.49) LCKEGFRALK
SCHEMBL18606983 0.84 LCK (0.51) LCKEGFRCDK4CCNA2CDK2
SCHEMBL18607342 0.84 ALK (0.44) LCKEGFRALKCCNA2CDK2
SCHEMBL20365609 0.82 EGFR (0.53) LCKEGFR
SCHEMBL18607343 0.81 EGFR (0.61) EGFR
SCHEMBL18607335 0.81 LCK (0.54) LCKEGFRCDK2
SCHEMBL18606898 0.80 LCK (0.45) LCKEGFRALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017035753-A1 2-ARYLAMINO PYRIDINE, PYRIDINE OR TRIAZINE DERIVATIVE, PREPARATION METHOD AND USE THEREOF 无锡双良生物科技有限公司 2017-03-09 WO disclosed