SCHEMBL18626319

SCHEMBL18626319

COc1cc([C@@H](C)C(C)C)ccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOX P28300 1/20 0.46
LOXL2 Q9Y4K0 1/20 0.46
KCNB1 Q14721 1/20 0.37
ROCK2 O75116 1/20 0.36
PFKFB3 Q16875 1/20 0.36
AAK1 Q2M2I8 4/20 0.35
CCR1 P32246 1/20 0.35
CCR5 P51681 1/20 0.35
CCR8 P51685 1/20 0.35
LRRK2 Q5S007 1/20 0.35
ACVR2A P27037 2/20 0.35
TGFBR2 P37173 2/20 0.35
ACACB O00763 1/20 0.35
DYRK1A Q13627 1/20 0.34
IDO1 P14902 1/20 0.34
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17000208 1.00 LOX (0.46) LOXLOXL2KCNB1ROCK2PFKFB3
SCHEMBL19863984 1.00 LOX (0.46) LOXLOXL2KCNB1ROCK2PFKFB3
SCHEMBL31421700 0.84 LOX (0.48) LOXLOXL2KCNB1ROCK2PFKFB3
SCHEMBL84460 0.84 LOX (0.48) LOXLOXL2KCNB1ROCK2PFKFB3
SCHEMBL22585542 0.83 LOX (0.44) LOXLOXL2KCNB1ROCK2PFKFB3
SCHEMBL12093566 0.82 LOX (0.47) LOXLOXL2KCNB1ROCK2PFKFB3
SCHEMBL17000210 0.81 ACACB (0.42) LOXLOXL2KCNB1ACACBGABRA1
SCHEMBL23232590 0.81 LOX (0.50) LOXLOXL2KCNB1ROCK2PFKFB3
SCHEMBL22369466 0.81 LOX (0.50) LOXLOXL2KCNB1ROCK2PFKFB3
SCHEMBL23232245 0.81 LOX (0.50) LOXLOXL2KCNB1ROCK2PFKFB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9593095-B2 Methods for the treatment of bacterial infections DUKE UNIVERSITY (US) 2017-03-14 US disclosed