SCHEMBL1862997

SCHEMBL1862997

O=C(NCCO)c1ccc(C(F)(F)F)c(-c2ccc3c(Nc4ccc(C(F)(F)F)cn4)ccnc3n2)n1

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 19/20 0.64
MAPK3 P27361 1/20 0.64
MAOA P21397 1/20 0.47
KCNH2 Q12809 1/20 0.47
SCN9A Q15858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12666839 0.90 TRPV1 (0.57) TRPV1MAPK3MAOAKCNH2SCN9A
SCHEMBL1865975 0.89 TRPV1 (0.67) TRPV1MAPK3MAOAKCNH2
SCHEMBL1858546 0.89 TRPV1 (0.62) TRPV1MAPK3SCN9A
SCHEMBL1863793 0.88 TRPV1 (0.64) TRPV1MAPK3MAOAKCNH2SCN9A
SCHEMBL1865075 0.88 TRPV1 (0.70) TRPV1MAPK3MAOAKCNH2
SCHEMBL1863481 0.87 TRPV1 (0.70) TRPV1MAPK3MAOAKCNH2
SCHEMBL1860025 0.87 TRPV1 (0.69) TRPV1MAPK3MAOAKCNH2
SCHEMBL1864308 0.87 TRPV1 (0.62) TRPV1MAPK3MAOAKCNH2
SCHEMBL1866310 0.85 TRPV1 (0.66) TRPV1MAPK3MAOAKCNH2
SCHEMBL1862099 0.84 TRPV1 (0.63) TRPV1MAPK3MAOAKCNH2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7935702-B2 Substituted biaryl quinolin-4-ylamine analogues NEUROGEN CORPORATION (US) 2011-05-03 US disclosed
US-7935702-B2 Substituted biaryl quinolin-4-ylamine analogues NEUROGEN CORPORATION (US) 2011-05-03 US disclosed