SCHEMBL18634646

SCHEMBL18634646

Cc1ncc(C)n2nc(CCc3nc4c5nccc(-c6nc(C)c7cc(CCc8nc9c%10ncccc%10sc9n8C)nn7c6C)c5ccc4n3C)cc12

nearest known ligand 0.42

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 13/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10309336 0.85 PDE10A (0.52) PDE10A
SCHEMBL10309348 0.79 PDE10A (0.54) PDE10A
SCHEMBL10309447 0.74 PDE10A (0.70) PDE10A
SCHEMBL10309354 0.73 PDE10A (0.52) PDE10A
SCHEMBL18634454 0.71 PDE10A (0.47) PDE10A
SCHEMBL18634565 0.69 PDE10A (0.66) PDE10A
SCHEMBL19965860 0.68 PDE10A (0.48) PDE10A
SCHEMBL10309340 0.64 PDE10A (0.59) PDE10A
SCHEMBL12066224 0.63 PDE10A (0.63) PDE10A
SCHEMBL10309383 0.62 PDE10A (0.63) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3210984-B1 HETEROARYL COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC (US) 2019-06-19 EP disclosed
EP-3210984-A1 HETEROARYL COMPOUNDS AND METHODS OF USE THEREOF Sunovion Pharmaceuticals Inc. (US) 2017-08-30 EP disclosed
EP-2663565-B1 HETEROARYL COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC (US) 2017-03-15 EP disclosed