SCHEMBL18634702

SCHEMBL18634702

CC(C)(C)OC(=O)[C@H](CCC1CC1)[C@@H](CCCC(F)(F)F)C(=O)OCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.44
POLB P06746 1/20 0.39
ITGB3 P05106 2/20 0.38
ITGA2B P08514 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
SYK P43405 1/20 0.38
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
LTA4H P09960 1/20 0.36
MAPT P10636 1/20 0.36
CTSL P07711 1/20 0.36
ABCB1 P08183 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18634622 0.93 AAK1 (0.43) AAK1POLBITGB3ITGA2BCYP3A4
SCHEMBL15626653 0.90 AAK1 (0.50) AAK1POLBSYKLTA4HMAPT
SCHEMBL15627206 0.88 AAK1 (0.45) AAK1POLBCYP3A4CYP2C9CYP2C19
SCHEMBL15627205 0.88 AAK1 (0.45) AAK1POLBCYP3A4CYP2C9CYP2C19
SCHEMBL15629455 0.87 AAK1 (0.47) AAK1POLBSYKLTA4HMAPT
SCHEMBL12690327 0.86 AAK1 (0.53) AAK1POLBSYKLTA4HMAPT
SCHEMBL16814420 0.84 AAK1 (0.47) AAK1POLBSYKLTA4HMAPT
SCHEMBL16983171 0.83 POLB (0.39) POLBCYP3A4CYP2C9CYP2C19SYK
SCHEMBL17263354 0.83 POLB (0.39) POLBCYP3A4CYP2C9CYP2C19SYK
SCHEMBL18634820 0.83 AAK1 (0.38) AAK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2897938-B1 FLUOROALKYL DIBENZODIAZEPINONE COMPOUNDS BRISTOL MYERS SQUIBB CO (US) 2017-03-15 EP disclosed