SCHEMBL18643545

SCHEMBL18643545

COc1cc2nc(C)[nH]c(=O)c2c(OC)c1CN1CCOCC1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.40
PARP1 P09874 1/20 0.40
TP53 P04637 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
PDE5A O76074 1/20 0.39
PDE11A Q9HCR9 1/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MAPK1 P28482 1/20 0.39
EZH2 Q15910 1/20 0.38
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
HSD17B10 Q99714 2/20 0.38
BRD4 O60885 1/20 0.38
SRC P12931 1/20 0.38
MAPT P10636 1/20 0.37
SYK P43405 1/20 0.37
HTT P42858 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21524670 0.87 PARP1 (0.38) PDE10APARP1TP53RXFP1PDE5A
SCHEMBL145199 0.84 BRD4 (0.47) PARP1TP53RXFP1BRD4MAPT
SCHEMBL30434436 0.84 BRD4 (0.47) PARP1TP53RXFP1BRD4MAPT
SCHEMBL30434906 0.82 PIK3CD (0.39) PDE10APARP1TP53RXFP1ALDH1A1
SCHEMBL30434568 0.81 BRD4 (0.54) PARP1BRD4
SCHEMBL121706 0.81 BRD4 (0.54) PARP1BRD4
Hydrochloric Acid SCHEMBL30434224 0.80 BRD4 (0.53) PARP1BRD4
Hydrochloric Acid SCHEMBL148595 0.80 BRD4 (0.53) PARP1BRD4
SCHEMBL349746 0.75 TP53 (0.40) PDE10APARP1TP53RXFP1PDE5A
SCHEMBL15302118 0.71 KDM1A (0.53) MAPK1SRCLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017041701-A1 NITRIC OXIDE-RELEASING PRODRUG MOLECULE 浙江华海药业股份有限公司 2017-03-16 WO disclosed