SCHEMBL18660566

SCHEMBL18660566

Nc1ncnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)c4ccccc4)c3F)c12

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 9/20 0.61
CYP2C19 P33261 9/20 0.51
CYP3A4 P08684 9/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12655324 0.82 CYP2C9 (0.58) CYP2C9CYP2C19CYP3A4
SCHEMBL1094221 0.79 CYP2C9 (0.66) CYP2C9CYP2C19CYP3A4
SCHEMBL1941592 0.79 BTK (0.69)
SCHEMBL287955 0.77 CYP2C9 (0.66) CYP2C9CYP2C19CYP3A4
SCHEMBL1093341 0.77 CYP2C9 (0.68) CYP2C9CYP2C19CYP3A4
SCHEMBL298822 0.77 CYP2C9 (0.75) CYP2C9CYP2C19CYP3A4
SCHEMBL292670 0.76 CYP2C9 (1.00) CYP2C9CYP2C19CYP3A4
SCHEMBL1817466 0.76 CYP2C19 (0.79) CYP2C9CYP2C19CYP3A4
SCHEMBL288245 0.75 CYP2C9 (0.63) CYP2C9CYP2C19CYP3A4
SCHEMBL1940319 0.74 BTK (0.59) CYP2C9CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2501236-B1 N-[2-fluoro-3-(4-amino-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-phenyl]-4-benzenesulfonamide derivatives as Raf protein kinase modulators for the treatment of cancer PLEXXIKON INC (US) 2017-03-29 EP disclosed