SCHEMBL1867213

SCHEMBL1867213

CCOC(=O)C1=CC2(CCC1S(=O)(=O)Nc1ccc(F)cc1Cl)OC[C@H]([C@H]1COC(C)(C)O1)O2

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 9/20 0.61
NPSR1 Q6W5P4 1/20 0.35
MRGPRX1 Q96LB2 4/20 0.34
LMNA P02545 2/20 0.34
KMT2A Q03164 1/20 0.33
HRH1 P35367 1/20 0.33
TSPO P30536 1/20 0.33
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12634741 0.90 TLR4 (0.65) TLR4MRGPRX1LMNAKMT2AHRH1
SCHEMBL1872797 0.89 TLR4 (0.62) TLR4NPSR1MRGPRX1LMNAKMT2A
SCHEMBL15146253 0.89 TLR4 (0.62) TLR4NPSR1MRGPRX1LMNAKMT2A
SCHEMBL1863349 0.89 TLR4 (0.62) TLR4NPSR1MRGPRX1LMNAKMT2A
SCHEMBL1863586 0.89 TLR4 (0.62) TLR4NPSR1MRGPRX1LMNAKMT2A
SCHEMBL4144992 0.89 TLR4 (0.46) TLR4MRGPRX1LMNAKMT2ATP53
SCHEMBL1865243 0.89 TLR4 (0.68) TLR4NPSR1MRGPRX1LMNAKMT2A
SCHEMBL1863271 0.88 TLR4 (0.65) TLR4NPSR1MRGPRX1LMNAKMT2A
SCHEMBL12634733 0.88 TLR4 (0.61) TLR4NPSR1MRGPRX1LMNAKMT2A
SCHEMBL1863576 0.87 TLR4 (0.68) TLR4NPSR1MRGPRX1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7935835-B2 Substituted cycloalkene derivative DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-05-03 US disclosed