SCHEMBL18680904

SCHEMBL18680904

CC(C)Nc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NSc4cccc(C#N)c4)c3F)c12

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 11/20 0.57
CYP2C9 P11712 8/20 0.57
CYP2C19 P33261 8/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18680611 0.91 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19
SCHEMBL18680683 0.90 CYP2C9 (0.66) CYP3A4CYP2C9CYP2C19
SCHEMBL18680699 0.88 CYP3A4 (0.62) CYP3A4CYP2C9CYP2C19
SCHEMBL18681124 0.85 CYP3A4 (0.72) CYP3A4CYP2C9CYP2C19
SCHEMBL18680843 0.85 CYP3A4 (0.62) CYP3A4CYP2C9CYP2C19
SCHEMBL1816626 0.84 CYP3A4 (0.74) CYP3A4CYP2C9CYP2C19
SCHEMBL18680654 0.84 CYP2C9 (0.60) CYP3A4CYP2C9CYP2C19
SCHEMBL18680733 0.83 CYP3A4 (0.61) CYP3A4CYP2C9CYP2C19
SCHEMBL18680905 0.83 CYP3A4 (0.62) CYP3A4CYP2C9CYP2C19
SCHEMBL18680694 0.82 CYP2C9 (0.71) CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2501236-B1 N-[2-fluoro-3-(4-amino-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-phenyl]-4-benzenesulfonamide derivatives as Raf protein kinase modulators for the treatment of cancer PLEXXIKON INC (US) 2017-03-29 EP disclosed