SCHEMBL18680974

SCHEMBL18680974

COc1ccc(S(=O)(=O)Nc2ccc(F)c(C(O)c3c[nH]c4ncnc(NCC5CC5)c34)c2F)cc1F

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 11/20 0.52
CYP2C19 P33261 8/20 0.41
CYP2C9 P11712 8/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18680881 0.89 CYP3A4 (0.55) CYP3A4CYP2C19CYP2C9
SCHEMBL1819345 0.84 CYP3A4 (0.74) CYP3A4CYP2C19CYP2C9
SCHEMBL16266429 0.81 CYP3A4 (0.45) CYP3A4
SCHEMBL12655351 0.76 CYP3A4 (0.71) CYP3A4CYP2C19CYP2C9
SCHEMBL1816704 0.75 CYP3A4 (0.82) CYP3A4CYP2C19CYP2C9
SCHEMBL2026944 0.74 CYP3A4 (0.75) CYP3A4CYP2C19CYP2C9
SCHEMBL1817568 0.74 CYP3A4 (0.77) CYP3A4CYP2C19CYP2C9
SCHEMBL1818232 0.73 CYP3A4 (0.67) CYP3A4CYP2C19CYP2C9
SCHEMBL18680973 0.73 CYP3A4 (0.78) CYP3A4CYP2C19CYP2C9
SCHEMBL1817438 0.72 CYP3A4 (0.77) CYP3A4CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2501236-B1 N-[2-fluoro-3-(4-amino-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-phenyl]-4-benzenesulfonamide derivatives as Raf protein kinase modulators for the treatment of cancer PLEXXIKON INC (US) 2017-03-29 EP disclosed