SCHEMBL18686209

SCHEMBL18686209

CCCc1ccc(NC(=O)c2c[nH]c3ccccc3c2=O)cc1NC(=O)O

nearest known ligand 0.75

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CFTR P13569 19/20 0.75
MAOB P27338 1/20 0.58
GABRA1 P14867 1/20 0.56
GABRB1 P18505 1/20 0.56
GABRA5 P31644 1/20 0.56
GABRA3 P34903 1/20 0.56
GABRA2 P47869 1/20 0.56
GABRB2 P47870 1/20 0.56
GABRA4 P48169 1/20 0.56
GABRA6 Q16445 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18686219 0.96 CFTR (0.72) CFTRMAOBGABRA1GABRB1GABRA5
SCHEMBL18686226 0.94 CFTR (0.77) CFTRMAOBGABRA1GABRB1GABRA5
SCHEMBL397792 0.91 CFTR (0.70) CFTRMAOBGABRA1GABRB1GABRA5
SCHEMBL398603 0.90 CFTR (0.72) CFTRMAOBGABRA1GABRB1GABRA5
SCHEMBL397397 0.90 CFTR (0.72) CFTRMAOBGABRA1GABRB1GABRA5
SCHEMBL18686214 0.90 CFTR (0.73) CFTRMAOBGABRA1GABRB1GABRA5
SCHEMBL399212 0.89 CFTR (0.70) CFTRMAOBGABRA1GABRB1GABRA5
SCHEMBL396591 0.88 CFTR (0.69) CFTRMAOBGABRA1GABRB1GABRA5
SCHEMBL397525 0.87 CFTR (0.71) CFTRMAOBGABRA1GABRB1GABRA5
SCHEMBL399222 0.87 CFTR (0.75) CFTRMAOBGABRA1GABRB1GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2502911-B1 Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2017-04-05 EP claimed