SCHEMBL18697237

SCHEMBL18697237

C=N/C(=C\C(=C/C)C(=O)NCc1n[nH]c2ccc(Cl)cc12)Cc1cc(C(N)=O)c2ncc(C)cc2c1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33
PARP1 P09874 1/20 0.32
KLKB1 P03952 2/20 0.32
CD38 P28907 2/20 0.32
KDR P35968 1/20 0.31
RPS6KB1 P23443 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18697211 0.83 KLKB1 (0.39) KLKB1
SCHEMBL18458953 0.81 KLKB1 (0.45) KLKB1
SCHEMBL20616373 0.80 KLKB1 (0.46) KLKB1
SCHEMBL23279872 0.79 KLKB1 (0.40) PARP1KLKB1
SCHEMBL17447329 0.76 KLKB1 (0.45) KLKB1
SCHEMBL18459038 0.76 KLKB1 (0.41) KLKB1
SCHEMBL17442701 0.76 KLKB1 (0.53) KLKB1
SCHEMBL20282946 0.71 KLKB1 (0.36) KLKB1
SCHEMBL21064331 0.71 KLKB1 (0.45) KLKB1
SCHEMBL17442728 0.69 KLKB1 (0.56) KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9611252-B2 Therapeutic inhibitory compounds LIFESCI PHARMACEUTICALS, INC. (BB) 2017-04-04 US disclosed