SCHEMBL1869908

SCHEMBL1869908

CCOC(=O)C1=CC2(CCC1S(=O)(=O)Nc1ccc(F)cc1Cl)O[C@@H](CNC(C)=O)[C@H](CNC(C)=O)O2

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 9/20 0.61
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37
LMNA P02545 2/20 0.36
TP53 P04637 1/20 0.36
MRGPRX1 Q96LB2 3/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
TSPO P30536 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HRH1 P35367 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1869905 1.00 TLR4 (0.61) TLR4PSEN1PSEN2APH1BNCSTN
SCHEMBL1866346 0.90 TLR4 (0.65) TLR4LMNATP53MRGPRX1KMT2A
SCHEMBL1862533 0.90 TLR4 (0.65) TLR4LMNATP53MRGPRX1KMT2A
SCHEMBL1866486 0.90 TLR4 (0.65) TLR4LMNATP53MRGPRX1KMT2A
SCHEMBL1862850 0.90 TLR4 (0.65) TLR4LMNATP53MRGPRX1KMT2A
SCHEMBL1862992 0.90 TLR4 (0.62) TLR4LMNATP53MRGPRX1KMT2A
SCHEMBL4159467 0.90 TLR4 (0.48) TLR4PSEN1PSEN2APH1BNCSTN
SCHEMBL1864585 0.89 TLR4 (0.63) TLR4LMNATP53MRGPRX1KMT2A
SCHEMBL1863029 0.89 TLR4 (0.63) TLR4LMNATP53MRGPRX1KMT2A
SCHEMBL1863576 0.88 TLR4 (0.68) TLR4LMNAMRGPRX1KMT2ATSPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7935835-B2 Substituted cycloalkene derivative DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-05-03 US disclosed
EP-1935879-A1 SUBSTITUTED CYCLOALKENE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2008-06-25 EP disclosed