SCHEMBL18707656

SCHEMBL18707656

C[C@@H]1C[C@@](c2cc(NC(=O)c3ncc(C#N)cc3Cl)ccc2F)(C(F)F)N=C(N)O1

nearest known ligand 0.69

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.69
BACE2 Q9Y5Z0 3/20 0.63
APP P05067 1/20 0.60
CYP3A4 P08684 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17119077 0.89 BACE1 (0.73) BACE1BACE2
SCHEMBL17119218 0.89 BACE1 (0.73) BACE1BACE2
SCHEMBL18707427 0.89 BACE1 (0.73) BACE1BACE2
SCHEMBL18708105 0.88 BACE1 (0.81) BACE1BACE2
SCHEMBL16918337 0.84 BACE1 (0.77) BACE1BACE2
SCHEMBL18707432 0.83 BACE1 (0.79) BACE1BACE2
SCHEMBL15345220 0.82 BACE1 (0.83) BACE1BACE2
SCHEMBL17119321 0.82 BACE1 (0.68) BACE1
SCHEMBL16041472 0.82 BACE1 (1.00) BACE1
SCHEMBL16042353 0.82 BACE1 (1.00) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9611261-B2 Perfluorinated cyclopropyl fused 1,3-oxazin-2-amine compounds as beta-secretase inhibitors and methods of use AMGEN INC. (US) 2017-04-04 US disclosed