SCHEMBL18733859

SCHEMBL18733859

Brc1cccc(CN2CCOc3ccccc3C2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
MBTD1 Q05BQ5 1/20 0.44
L3MBTL3 Q96JM7 1/20 0.44
CYP2D6 P10635 1/20 0.44
KDM4E B2RXH2 1/20 0.43
FAAH O00519 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
APP P05067 1/20 0.42
CLPP Q16740 1/20 0.41
PTGER2 P43116 1/20 0.41
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6436620 0.84 CYP2D6 (0.51) CYP2D6APPHTR1A
SCHEMBL3277742 0.83 CYP2D6 (0.48) CYP2D6MEN1KMT2APTGER2DRD2
SCHEMBL3276408 0.83 CYP2D6 (0.51) CYP2D6MEN1KMT2APTGER2DRD2
SCHEMBL18734068 0.80 PTGER2 (0.52) CYP2D6APPPTGER2SIRT2HTR1A
SCHEMBL22512823 0.79 MEN1 (0.44) TDP1KDM4EMEN1KMT2AAPP
SCHEMBL12451410 0.76 CYP1A2 (0.51) SMN1; SMN2TDP1CYP2D6KDM4EHTR1A
SCHEMBL578335 0.75 SMN1; SMN2 (0.70) SMN1; SMN2TDP1MBTD1L3MBTL3KDM4E
SCHEMBL18706621 0.74 SIRT2 (0.44) SMN1; SMN2TDP1MBTD1L3MBTL3KDM4E
SCHEMBL18706622 0.74 SIRT2 (0.44) SMN1; SMN2TDP1MBTD1L3MBTL3KDM4E
SCHEMBL17160816 0.74 SMN1; SMN2 (0.68) SMN1; SMN2TDP1MBTD1L3MBTL3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017060854-A1 BIARYL PYRAZOLES AS NRF2 REGULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-04-13 WO disclosed