SCHEMBL18740465

SCHEMBL18740465

CCCN(CCC)S(=O)(=O)c1cccc(C(=O)N[C@@H](Cc2cc(F)cc(F)c2)[C@H](O)CNCc2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.60
BACE2 Q9Y5Z0 11/20 0.60
CTSD P07339 10/20 0.60
CTSB P07858 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13306832 0.92 BACE1 (0.68) BACE1BACE2CTSDCTSB
SCHEMBL3351108 0.92 BACE1 (0.68) BACE1BACE2CTSDCTSB
SCHEMBL3351111 0.92 BACE1 (0.68) BACE1BACE2CTSDCTSB
SCHEMBL18740514 0.92 BACE1 (0.59) BACE1BACE2CTSDCTSB
SCHEMBL18740470 0.91 BACE1 (0.57) BACE1BACE2CTSDCTSB
SCHEMBL18740509 0.86 BACE1 (0.68) BACE1BACE2CTSD
SCHEMBL18767148 0.86 BACE1 (0.78) BACE1BACE2CTSD
SCHEMBL18740491 0.85 BACE1 (0.60) BACE1BACE2CTSDCTSB
SCHEMBL3353685 0.85 BACE1 (0.69) BACE1BACE2CTSDCTSB
SCHEMBL3353677 0.85 BACE1 (0.69) BACE1BACE2CTSDCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017066742-A1 BACE-2 INHIBITORY COMPOUNDS AND RELATED METHODS OF USE JORTAN PHARMACEUTICALS INC. (US) 2017-04-20 WO disclosed