SCHEMBL18751647

SCHEMBL18751647

CNC(=O)c1c(-c2ccc(F)cc2)oc2ccc(-c3cc(C(N)=O)ccc3C)c(F)c12

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 6/20 0.67
KCNH2 Q12809 3/20 0.67
CYP3A4 P08684 5/20 0.51
NR1I2 O75469 1/20 0.48
APP P05067 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14217296 0.91 KCNH2 (0.68) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL142336 0.91 KCNH2 (0.68) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL9919844 0.89 CYP2C8 (0.66) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL18752213 0.87 CYP2C8 (0.55) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL12447856 0.84 KCNH2 (0.60) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL10242360 0.83 CYP2C8 (0.58) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL1919345 0.83 CYP2C8 (0.58) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL18751750 0.82 CYP2C8 (0.52) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL1919338 0.82 CYP2C8 (0.57) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL2141860 0.81 CYP2C8 (0.84) CYP2C8KCNH2CYP3A4NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545051-B1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2017-04-19 EP disclosed