SCHEMBL18759307

SCHEMBL18759307

CCC(O)CS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(-c4ccc(Cl)cc4)cc23)c1F

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 4/20 0.83
RIPK2 O43353 2/20 0.83
RAF1 P04049 2/20 0.83
KDR P35968 2/20 0.83
MAP2K2 P36507 2/20 0.83
TGFBR2 P37173 2/20 0.83
NEK2 P51955 2/20 0.83
MAP2K1 Q02750 2/20 0.83
TNK2 Q07912 2/20 0.83
MAP2K5 Q13163 2/20 0.83
PTK6 Q13882 2/20 0.83
NEK11 Q8NG66 2/20 0.83
MAP3K20 Q9NYL2 2/20 0.83
MAP4K5 Q9Y4K4 2/20 0.83
ABCB11 O95342 1/20 0.83
EGFR P00533 1/20 0.83
KRAS P01116 1/20 0.83
PGR P06401 1/20 0.83
RET P07949 1/20 0.83
CHRM2 P08172 1/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18759119 0.94 BRAF (0.78) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL20399953 0.93 BRAF (0.79) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL20399246 0.93 BRAF (0.79) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL18759294 0.93 BRAF (0.79) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL298547 0.92 BRAF (0.80) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL7876722 0.92 BRAF (0.89) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL12891936 0.91 BRAF (1.00) BRAFRIPK2RAF1KDRMAP2K2
Vemurafenib SCHEMBL29355460 0.91 BRAF (1.00) BRAFRIPK2RAF1KDRMAP2K2
Vemurafenib SCHEMBL29356185 0.91 BRAF (1.00) BRAFRIPK2RAF1KDRMAP2K2
Vemurafenib SCHEMBL298931 0.91 BRAF (1.00) BRAFRIPK2RAF1KDRMAP2K2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017066193-A1 NOVEL INHIBITORS OF PROTEIN KINASES PRINCETON DRUG DISCOVERY, LLC (US) 2017-04-20 WO disclosed