SCHEMBL18769435

SCHEMBL18769435

NNC1OC1c1cnc(NC2(c3cccc(C(F)(F)F)c3)CC2)nc1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 13/20 0.57
HDAC3 O15379 6/20 0.57
HDAC1 Q13547 6/20 0.57
HDAC2 Q92769 6/20 0.57
VNN1 O95497 3/20 0.51
KDM1A O60341 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24968633 0.78 HDAC6 (0.67) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL28247594 0.78 HDAC6 (0.66) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL18742382 0.76 HDAC6 (0.82) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL28247610 0.74 HDAC6 (0.61) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL28248169 0.73 HDAC6 (0.60) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL4729657 0.73 HDAC3 (1.00) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL18742434 0.72 HDAC6 (0.78) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL22804912 0.72 HDAC6 (0.60) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL29581928 0.72 HDAC6 (0.60) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL18742577 0.72 HDAC3 (0.75) HDAC6HDAC3HDAC1HDAC2VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017065473-A1 OXADIAZOLE AMINE DERIVATIVE COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND THE PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2017-04-20 WO disclosed