SCHEMBL18790871

SCHEMBL18790871

CC1(C)OC2=C(C(=O)c3ccccc3C2=O)C1Br

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 16/20 0.68
NQO1 P15559 2/20 0.43
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
POLB P06746 2/20 0.40
KDM4E B2RXH2 1/20 0.39
CES2 O00748 1/20 0.39
GMNN O75496 1/20 0.39
TDP2 O95551 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
GLA P06280 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
HSPD1 P10809 1/20 0.39
THRB P10828 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13443011 0.81 IDO1 (1.00) IDO1NQO1
SCHEMBL13443001 0.81 IDO1 (1.00) IDO1NQO1
SCHEMBL13443002 0.79 IDO1 (1.00) IDO1NQO1MEN1KMT2AKDM4E
SCHEMBL3618661 0.79 IDO1 (1.00) IDO1NQO1MEN1KMT2AKDM4E
SCHEMBL18791132 0.76 IDO1 (0.56) IDO1NQO1MEN1KMT2APOLB
SCHEMBL13443005 0.74 IDO1 (1.00) IDO1NQO1MEN1KMT2APOLB
SCHEMBL14069791 0.74 IDO1 (0.69) IDO1NQO1
SCHEMBL3616835 0.74 IDO1 (1.00) IDO1NQO1MEN1KMT2APOLB
SCHEMBL13443009 0.74 IDO1 (1.00) IDO1NQO1MEN1KMT2APOLB
SCHEMBL18791133 0.73 IDO1 (0.63) IDO1NQO1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017070012-A1 LAPACHONE DERIVATIVES CONTAINING TWO REDOX CENTERS AND METHODS OF USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2017-04-27 WO disclosed