SCHEMBL18809192

SCHEMBL18809192

CNC(=O)c1c(-c2ccc(F)cc2)oc2nc(NCC(F)F)c(-c3ccc(F)c(C(=O)NC45CCC(C4)C5)c3)cc12

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.37
CYP2C8 P10632 4/20 0.36
KCNH2 Q12809 2/20 0.36
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
NR1I2 O75469 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16114410 0.94 CYP3A4 (0.39) CYP3A4CYP2C8KCNH2CNR1CNR2
SCHEMBL18809269 0.92 CYP3A4 (0.36) CYP3A4CYP2C8KCNH2CNR1CNR2
SCHEMBL17466568 0.90 CYP3A4 (0.39) CYP3A4CYP2C8KCNH2
SCHEMBL16133737 0.86 CYP3A4 (0.37) CYP3A4CYP2C8KCNH2CNR1CNR2
SCHEMBL16113837 0.85 CYP3A4 (0.42) CYP3A4CYP2C8
SCHEMBL16133450 0.84 CYP3A4 (0.43) CYP3A4CYP2C8KCNH2CNR1CNR2
SCHEMBL16133784 0.84 CYP2C8 (0.41) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL17466585 0.83 CYP3A4 (0.38) CYP3A4CYP2C8KCNH2CNR1CNR2
SCHEMBL17466567 0.82 CYP3A4 (0.38) CYP3A4CYP2C8KCNH2
SCHEMBL18809609 0.81 CYP3A4 (0.40) CYP3A4CYP2C8KCNH2NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970174-B1 FUSED FURANS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2017-05-03 EP disclosed