SCHEMBL18809558

SCHEMBL18809558

CNC(O)c1c(-c2ccc(F)cc2)oc2cc([N+](=O)[O-])c(-c3cc(C(=O)NC45CC(C4)C5)c(F)cc3F)cc12

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 4/20 0.33
CNR1 P21554 3/20 0.33
ALDH1A1 P00352 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
SCN9A Q15858 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PAX8 Q06710 1/20 0.32
THRA P10827 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17453371 0.88 CYP3A4 (0.40)
SCHEMBL16112908 0.75 CYP3A4 (0.42)
SCHEMBL16112897 0.73 CYP3A4 (0.41)
SCHEMBL16133453 0.73 CNR1 (0.40) CNR2CNR1
SCHEMBL19309893 0.72 MAPT (0.33) ALDH1A1MEN1KMT2A
SCHEMBL16113159 0.72 CYP3A4 (0.38)
SCHEMBL16133806 0.72 CYP3A4 (0.40)
SCHEMBL18809559 0.71 CYP3A4 (0.36)
SCHEMBL18809631 0.70 CYP3A4 (0.43) CNR2CNR1
SCHEMBL16133773 0.67 CYP3A4 (0.42) CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970174-B1 FUSED FURANS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2017-05-03 EP disclosed