Temocapril

Temocapril

SCHEMBL188165

CCOC(=O)[C@H](CCc1ccccc1)N[C@H]1CS[C@H](c2cccs2)CN(CC(=O)O)C1=O

nearest known ligand 0.82

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACE P12821 6/20 0.54
ABCB11 O95342 1/20 0.54
AGTR2 P50052 1/20 0.54
PDE3A Q14432 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
KDM4E B2RXH2 1/20 0.53
CYP3A4 P08684 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Temocapril SCHEMBL10377817 1.00 ACE (0.54) ACEABCB11AGTR2PDE3ATDP1
Temocapril SCHEMBL6506860 1.00 ACE (0.54) ACEABCB11AGTR2PDE3ATDP1
Temocapril SCHEMBL10376961 1.00 ACE (0.54) ACEABCB11AGTR2PDE3ATDP1
Temocapril SCHEMBL1650365 1.00 ACE (0.54) ACEABCB11AGTR2PDE3ATDP1
Temocapril SCHEMBL6444389 1.00 ACE (0.54) ACEABCB11AGTR2PDE3ATDP1
Temocapril SCHEMBL10377818 1.00 ACE (0.54) ACEABCB11AGTR2PDE3ATDP1
Temocapril SCHEMBL10377820 1.00 ACE (0.54) ACEABCB11AGTR2PDE3ATDP1
Temocapril SCHEMBL121391 0.99 KDM4E (0.55) ACEABCB11AGTR2PDE3ATDP1
Temocapril SCHEMBL10431733 0.99 KDM4E (0.55) ACEABCB11AGTR2PDE3ATDP1
Temocapril SCHEMBL10431734 0.99 KDM4E (0.55) ACEABCB11AGTR2PDE3ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7022 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026087680-A1 TREATMENT FOR CARDIOVASCULAR DISEASE SAPREME TECHNOLOGIES B.V. (NL) 2026-04-30 WO claimed
EP-4595974-A2 THERAPEUTIC COMBINATIONS OF TDFRPS AND ADDITIONAL AGENTS AND METHODS OF USE Carlson, William D. (US) 2025-08-06 EP claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
US-20250082608-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE SINGAPORE HEALTH SERVICES PTE LTD. (SG) 2025-03-13 US claimed
US-12194032-B2 Method of treating focal segmental glomerulosclerosis CHEMOCENTRYX, INC. (US) 2025-01-14 US claimed
US-20240374587-A1 MEDICINE FOR PREVENTION AND TREATMENT OF DISEASES LINKED TO ANTI-OBESITY ACTIVITY SHIONOGI & CO., LTD. (JP) 2024-11-14 US claimed
EP-4134080-B1 CCR2 INHIBITORS FOR USE IN TREATING RENAL DISEASES CHEMOCENTRYX INC (US) 2024-11-13 EP claimed
EP-4448096-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE Singapore Health Services Pte. Ltd. (SG) 2024-10-23 EP claimed
WO-2024210922-A1 COMPOSITIONS FOR ANTIHYPERTENSIVE DRUGS INNOVATOR THERAPEUTICS, LLC. (US) 2024-10-10 WO claimed
EP-3083573-B1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME LLC (US) 2024-08-07 EP claimed
EP-0808171-A2 COMBINATION OF ANGIOTENSIN CONVERTING ENZYME INHIBITOR, SIDE-EFFECT-REDUCED AMOUNT OF ALDOSTERONE ANTAGONIST AND DIURETIC G.D. SEARLE & CO. (US) 1997-11-26 EP claimed
EP-0808172-A2 COMBINATION OF ANGIOTENSIN CONVERTING ENZYME INHIBITOR AND SIDE-EFFECT-REDUCED AMOUNT OF ALDOSTERONE ANTAGONIST G.D. SEARLE & COMPANY (US) 1997-11-26 EP claimed
WO-1997002032-A1 METHOD OF TREATING RENAL DISEASE USING AN ACE INHIBITOR AND AN AII ANTAGONIST MERCK & CO., INC. (US) 1997-01-23 WO claimed
WO-1996024372-A2 COMBINATION OF ANGIOTENSIN CONVERTING ENZYME INHIBITOR, SIDE-EFFECT-REDUCED AMOUNT OF ALDOSTERONE ANTAGONIST AND DIURETIC G.D. SEARLE & CO. (US) 1996-08-15 WO claimed
WO-1996024373-A2 COMBINATION OF ANGIOTENSIN CONVERTING ENZYME INHIBITOR AND SIDE-EFFECT-REDUCED AMOUNT OF ALDOSTERONE ANTAGONIST G.D. SEARLE & CO. (US) 1996-08-15 WO claimed
EP-0643580-A4 COMBINATIONS OF ACE INHIBITORS AND DIURETICS. 1995-04-19 EP claimed
EP-0643580-A1 COMBINATIONS OF ACE INHIBITORS AND DIURETICS MERCK & CO. INC. (US) 1995-03-22 EP claimed
WO-1994028924-A1 COMBINATION OF ANGIOTENSIN CONVERTING ENZYME INHIBITORS AND AII ANTAGONISTS LABORATOIRES MERCK SHARP ET DOHME CHIBRET (FR) 1994-12-22 WO claimed
EP-0629408-A1 Combination of angiotensin converting enzyme inhibitors and AII antagonists LABORATOIRES MERCK, SHARP & DOHME-CHIBRET (FR) 1994-12-21 EP claimed
WO-1993017685-A1 COMBINATIONS OF ACE INHIBITORS AND DIURETICS MERCK & CO., INC. (US) 1993-09-16 WO claimed