SCHEMBL18818488

SCHEMBL18818488

CC(C)(C)OC(=O)N1Cc2cnc(O)nc2C1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.53
CRBN Q96SW2 1/20 0.53
MAPT P10636 2/20 0.52
NR1H2 P55055 2/20 0.44
ESR2 Q92731 1/20 0.44
HSP90AA1 P07900 3/20 0.40
MAPK1 P28482 1/20 0.40
HSP90B1 P14625 1/20 0.40
HDAC1 Q13547 1/20 0.39
CKS1B P61024 1/20 0.39
SKP1 P63208 1/20 0.39
SKP2 Q13309 1/20 0.39
GPR119 Q8TDV5 2/20 0.38
ROCK2 O75116 1/20 0.38
NAMPT P43490 2/20 0.38
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25574538 0.88 MAPT (0.67) DDB1CRBNMAPTNR1H2ESR2
SCHEMBL30378007 0.88 MAPT (0.67) DDB1CRBNMAPTNR1H2ESR2
SCHEMBL20078108 0.86 DDB1 (0.53) DDB1CRBNMAPTNR1H2ESR2
SCHEMBL17184636 0.85 DDB1 (0.53) DDB1CRBNMAPTNR1H2ESR2
SCHEMBL15875047 0.85 DDB1 (0.53) DDB1CRBNMAPTNR1H2ESR2
SCHEMBL11929937 0.85 DDB1 (0.55) DDB1CRBNMAPTNR1H2ESR2
SCHEMBL18570958 0.85 DDB1 (0.53) DDB1CRBNMAPTNR1H2ESR2
SCHEMBL740206 0.84 DDB1 (0.53) DDB1CRBNMAPTNR1H2ESR2
SCHEMBL13028051 0.84 DDB1 (0.52) DDB1CRBNMAPTNR1H2ESR2
SCHEMBL741949 0.83 CCNA2 (0.53) DDB1CRBNMAPTNR1H2ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107428762-B Phthalazinone derivatives, preparation method and use thereof 四川科伦博泰生物医药股份有限公司 2020-03-10 CN disclosed
WO-2017071636-A1 PHTHALAZINE KETONE DERIVATIVE, AND PREPARATION METHOD AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-05-04 WO disclosed