SCHEMBL18819035

SCHEMBL18819035

CN(c1ncc2c(n1)CNC2)C1CC1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.35
IRAK4 Q9NWZ3 2/20 0.34
MAPK10 P53779 1/20 0.31
JAK1 P23458 1/20 0.31
JAK3 P52333 1/20 0.31
HTR2C P28335 1/20 0.31
PDE10A Q9Y233 2/20 0.30
EHMT2 Q96KQ7 1/20 0.30
EHMT1 Q9H9B1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28413259 0.98 DYRK1A (0.34) DYRK1AIRAK4MAPK10JAK1JAK3
SCHEMBL18536681 0.84 GBA1 (0.36) IRAK4MAPK10HTR2C
SCHEMBL2809677 0.82 HSD17B10 (0.36) HTR2C
Hydrochloric Acid SCHEMBL28410160 0.80 HSD17B10 (0.35) HTR2C
SCHEMBL1528492 0.69 HTR2C (0.37) HTR2C
SCHEMBL1528578 0.68 HTR2C (0.34) HTR2C
SCHEMBL785776 0.68 POLB (0.48) HTR2C
SCHEMBL18818630 0.68 GRM5 (0.46) MAPK10
Hydrochloric Acid SCHEMBL2874635 0.67 HTR2C (0.36) HTR2C
Hydrochloric Acid SCHEMBL16060483 0.67 HTR2C (0.33) HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017071636-A1 PHTHALAZINE KETONE DERIVATIVE, AND PREPARATION METHOD AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-05-04 WO disclosed