SCHEMBL18833136

SCHEMBL18833136

CNc1c[nH]nc1-c1nc2cc(F)c(OCCN3CCCCC3)cc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.43
CHEK2 O96017 2/20 0.38
FGFR1 P11362 2/20 0.38
FLT1 P17948 2/20 0.38
LTA4H P09960 1/20 0.37
RUNX1 Q01196 2/20 0.37
BRD4 O60885 1/20 0.35
IL17A Q16552 1/20 0.35
CCR2 P41597 1/20 0.35
HRH4 Q9H3N8 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
IKBKE Q14164 1/20 0.34
TBK1 Q9UHD2 1/20 0.34
KDR P35968 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3926346 0.86 CHEK2 (0.41) ACHECHEK2FGFR1FLT1RUNX1
Hydrochloric Acid SCHEMBL4126862 0.85 CHEK2 (0.40) ACHECHEK2FGFR1FLT1RUNX1
SCHEMBL4133817 0.85 SYK (0.50) ACHECHEK2FGFR1FLT1KDR
Trifluoroacetic Acid SCHEMBL4129766 0.81 SYK (0.46) ACHECHEK2RUNX1TBK1KDR
SCHEMBL4142555 0.81 SYK (0.49) ACHECHEK2FGFR1FLT1HRH4
SCHEMBL18832926 0.81 HRH4 (0.37) ACHECHEK2HRH4
Hydrochloric Acid SCHEMBL4134722 0.80 SYK (0.49) CHEK2FGFR1FLT1HRH4KDR
SCHEMBL3924905 0.78 CHEK2 (0.39) CHEK2FGFR1FLT1KDR
SCHEMBL4133840 0.77 SYK (0.53) ACHECHEK2FGFR1FLT1HRH4
SCHEMBL13373931 0.76 SYK (0.45) HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041119-B1 PYRAZOLYLBENZIMIDAZOLE DERIVATIVES, COMPOSITIONS CONTAINING THEM AND USE THEREOF AVENTIS PHARMA SA (FR) 2017-05-10 EP disclosed