SCHEMBL18834052

SCHEMBL18834052

Cc1nc2c(c(=O)[nH]c(=O)n2C)n1Cc1ccc(Cl)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.72
APOBEC3G Q9HC16 1/20 0.72
TSHR P16473 8/20 0.69
ALDH1A1 P00352 7/20 0.69
MEN1 O00255 5/20 0.69
KMT2A Q03164 5/20 0.69
HPGD P15428 5/20 0.69
MAPK1 P28482 3/20 0.69
POLB P06746 3/20 0.68
TP53 P04637 2/20 0.64
XBP1 P17861 2/20 0.64
HSD17B10 Q99714 5/20 0.61
GAA P10253 1/20 0.61
DCTPP1 Q9H773 1/20 0.61
MAPT P10636 2/20 0.60
KDM1A O60341 1/20 0.60
BRAF P15056 2/20 0.58
USP2 O75604 2/20 0.58
BRDT Q58F21 1/20 0.58
GLA P06280 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6348692 0.88 BRAF (0.72) TSHRALDH1A1MEN1KMT2AMAPK1
SCHEMBL16028621 0.86 ATM (0.71) ATMAPOBEC3GTSHRALDH1A1MEN1
SCHEMBL19375412 0.86 ATM (0.71) ATMAPOBEC3GTSHRALDH1A1MEN1
SCHEMBL16028820 0.86 ATM (0.71) ATMAPOBEC3GTSHRALDH1A1MEN1
SCHEMBL16028236 0.83 ATM (0.67) ATMAPOBEC3GTSHRALDH1A1MEN1
SCHEMBL16028826 0.82 TSHR (1.00) ATMAPOBEC3GTSHRALDH1A1MEN1
SCHEMBL20652970 0.82 ATM (0.62) ATMAPOBEC3GTSHRALDH1A1MEN1
SCHEMBL16028896 0.80 TSHR (0.84) ATMAPOBEC3GTSHRALDH1A1MEN1
SCHEMBL5075029 0.80 POLB (0.84) ATMAPOBEC3GTSHRALDH1A1MEN1
SCHEMBL16028495 0.80 TSHR (0.67) ATMAPOBEC3GTSHRALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970303-B3 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES INC (US) 2018-08-01 EP disclosed
EP-2970303-B9 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES INC (US) 2017-09-20 EP disclosed
EP-2970303-B1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES INC (US) 2017-05-10 EP disclosed